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GBR-12909 2HCl

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Dopamine reuptake inhibitor CAS#: 67469-78-7 Citations: 1) Andersen et al. (1989), The dopamine inhibitor GBR 12909: selectivity and molecular mechanism of action; Eur. J. Pharmacol., 166 493 2) Contreras et al. (1990), GBR-12909 and fluspirilene potently inhibited binding of [3H] (+)3-PPP to sigma receptors in rat brain; Life Sci., 47 PL133 3) Yorgason et al. (2011), Low and high affinity dopamine transporter inhibitors block dopamine uptake within 5 sec of intravenous injection; Neuroscience, 182 125

Product Code: ax43825 (10 mg)

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Product Specification

Function / pharmacology Potent and selective inhibitor of dopamine reuptake (Ki = 1 nM) with greater than 100 fold selectivity over serotonin and noradrenaline1. Also acts as a potent sigma receptor ligand2. Very fast acting via i.v. administration3.
Chemical name 1-[2-[Bis-(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine dihydrochloride
Molecular weight 523.5
Molecular formula C28 H32 F2 N2 O · 2HCl
Physical description White solid
Solubility DMSO (30 mg/ml) Water (10 mg/ml)
Size 10 mg
Stability Stable for 2 years as supplied. Solutions in DMSO or distilled water may be stored at -20°C for up to 1 month.